✦ LIBER ✦

Binding of (+)PHNO and other D2-dopamine agonists to D1-dopamine receptors labelled by [3H]SCH 23390

✍ Scribed by D. J. Pettibone; J. A. Totaro; B. V. Clineschmidt

Publisher: Springer
Year: 1987
Tongue: English
Weight: 239 KB
Volume: 69
Category: Article
ISSN: 1435-1463
DOI: 10.1007/bf01244105

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Differential modulation of dopamine D1-r

Differential modulation of dopamine D1-receptor binding and mRNA expression in the basal ganglia by the D1-receptor antagonist, SCH-23390

✍ Jiang Yu; Héctor Coirini; Lillemor Källström; Frits-Axel Wiesel; Allan E. Johnso 📂 Article 📅 1998 🏛 John Wiley and Sons 🌐 English ⚖ 333 KB 👁 2 views

Dopamine D 1 -receptor binding in the basal ganglia is differentially regulated by subtype nonspecific dopamine antagonists such as the antipsychotic, Fluphenazine. The purpose of the present study was to determine the relative contributions of D 1 and D 2 receptor systems in the regulation of basal

Radiosynthesis of a selective dopamine D

Radiosynthesis of a selective dopamine D-1 receptor antagonist: R(+)-7-chloro-8-hydroxy-3-[11C]methyl-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine ([11C]SCH 23390)

✍ Hayden T. Ravert; Alan A. Wilson; Robert F. Dannals; Dean F. Wong; Henry N. Wagn 📂 Article 📅 1987 🏛 Elsevier Science ⚖ 200 KB

Carbon-11 labeled SCH 23390, a selective dopamine D-1 receptor antagonist (Fig. 1b), was prepared by N-alkylation of the nor-methyl precursor with [11C]iodomethane. The product was purified by semi-preparative HPLC and shown to be radiochemically pure at the end of synthesis. The synthesis was compl

ChemInform Abstract: cis- and trans-2,3,

ChemInform Abstract: cis- and trans-2,3,3a,4,5,9b-Hexahydro-1H-benz[e]indoles: Synthesis and Evaluation of Dopamine D2 and D3 Receptor Binding Affinity.

✍ Xiaodong Song; A. Michael Crider; Sharon F. Cruse; Debasis Ghosh; Cheryl Klein-S 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 40 KB 👁 1 views

fused pyrrole derivatives fused pyrrole derivatives R 0160 3,3a,4,5,indoles: Synthesis and Evaluation of Dopamine D 2 and D 3 Receptor Binding Affinity. -In order to find more D 3 receptor binding selective compounds different kinds of the title substances such as (X), (XI), and (XVIII) are synthes

Synthesis and evaluation of cis-1-methyl

Synthesis and evaluation of cis-1-methyl-3-n-propyl-2,3,3a,4,5,9b-hexahydro-1H-benz[e]indoles for in vitro dopamine D1 and D2 receptor binding affinity

✍ D Ghosh; C.L. Klein; B Garner; P.H. Andersen; A.M. Crider 📂 Article 📅 1995 🏛 Elsevier Science 🌐 French ⚖ 525 KB

18F-labeled benzamide derivatives: Synth

18F-labeled benzamide derivatives: Synthesis of 3,5-dichloro-N-[1-{2-[18F]-fluoroethyl}-2-pyrrolidinyl)methyl]-6-methoxysalicylamide And derivatives as dopamine D-2 receptor-binding radioligands

✍ N. Satyamurthy; J.R. Barrio; G.T. Bida; M.E. Phelps 📂 Article 📅 1989 🏛 John Wiley and Sons 🌐 French ⚖ 121 KB

Agonist and antagonist actions of yohimb

Agonist and antagonist actions of yohimbine as compared to fluparoxan at α2-adrenergic receptors (AR)s, serotonin (5-HT)1A, 5-HT1B, 5-HT1D and dopamine D2 and D3 receptors. Significance for the modulation of frontocortical monoaminergic transmission and depressive states

✍ Mark J. Millan; Adrian Newman-Tancredi; Valérie Audinot; Didier Cussac; François 📂 Article 📅 2000 🏛 John Wiley and Sons 🌐 English ⚖ 340 KB 👁 1 views

Herein, we evaluate the interaction of the ␣ 2 -AR antagonist, yohimbine, as compared to fluparoxan, at multiple monoaminergic receptors and examine their roles in the modulation of adrenergic, dopaminergic and serotonergic transmission in freelymoving rats. Yohimbine displays marked affinity at hum