## Abstract The synthesis of a series of 1‐aminoalkyl‐2‐benzyl‐nitro‐benzimidazoles is described. Many of the 5‐nitro‐benzimidazoles prepared show strong analgesic activity. 1‐(β‐Diethylamino‐ethyl)‐2‐(p‐ethoxy‐benzyl)‐5‐nitro‐benzimidazole (XXXVIII) is 1000 times as potent as morphine and therefor
Benzimidazol-Derivate und verwandte Heterocyclen. II. Synthese von 1-Aminoalkyl-2-benzyl-benzimidazolen
✍ Scribed by A. Hunger; J. Kebrle; A. Rossi; K. Hoffmann
- Publisher
- John Wiley and Sons
- Year
- 1960
- Tongue
- German
- Weight
- 655 KB
- Volume
- 43
- Category
- Article
- ISSN
- 0018-019X
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✦ Synopsis
Abstract
The synthesis of a series of 1‐aminoalkyl‐2‐benzyl‐benzimidazoles is described. Some of these compounds show strong analgesic activity.
📜 SIMILAR VOLUMES
## Abstract The synthesis of a series of phenyl‐[1‐aminoalkyl‐benzimidazolyl‐(2)]‐acetic esters and amides is described. Some of the derivatives prepared show pronounced analgesic activity.
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