Asymmetric synthesis of S-(+)-4-amino-5-hexynoic acid
β Scribed by Helena McAlonan; Paul J. Stevenson
- Publisher
- Elsevier Science
- Year
- 1995
- Tongue
- English
- Weight
- 410 KB
- Volume
- 6
- Category
- Article
- ISSN
- 0957-4166
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π SIMILAR VOLUMES
In an earlier communloatlon 1) , aaymmetrlc alkylatlon of cyclohexanone enamine wae described. Thle paper deale with an extenelon of thle reaction to the aldehyde enamlne. mamine alkylatlon was devleed by stork and hle co-workers 8)
Asymmetric synthesis of (+)-phosphinothricin, (+)-2-amino-4-phosphonobutyric acid, and their enantiomers has been achieved by the Michael addition of chiral glycine Schiff bases to vinyl phosphorus compounds. Phosphorus analogues of glutamic acid are interesting as biologically active substances. Th
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An asymmetric synthesis of (2S,4R)-4-hydroxypipecolic acid was accomplished in eight steps and 31% overall yield.