An efficient, convergent synthesis of an LTD 4 antagonist, RG12525 (1) has been achieved through the alkylation of the (2-quinolinylmethoxy)phenol (2) with either a triphenylmethyl protected tetrazole synthon (4a) or with a tetrahydropyranyl derivative (4b). Preparation of synthons 4a and 4b, as wel
โฆ LIBER โฆ
An efficient synthesis of LTD4 antagonist L-699,392
โ Scribed by King, A. O.; Corley, E. G.; Anderson, R. K.; Larsen, R. D.; Verhoeven, T. R.; Reider, P. J.; Xiang, Y. B.; Belley, M.; Leblanc, Y.
- Book ID
- 115504110
- Publisher
- American Chemical Society
- Year
- 1993
- Tongue
- English
- Weight
- 663 KB
- Volume
- 58
- Category
- Article
- ISSN
- 0022-3263
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