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A new versatile linker for the solid-phase synthesis of secondary amines

โœ Scribed by Heiko Glatz; Willi Bannwarth

Publisher
Elsevier Science
Year
2003
Tongue
French
Weight
238 KB
Volume
44
Category
Article
ISSN
0040-4039

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โœฆ Synopsis

A novel linker for the solid-phase synthesis of secondary amines based on an intramolecular cyclization was developed. The linker allows for a stepwise built-up of the secondary amines on the support. The feasibility was demonstrated in the parallel synthesis of a small set of different secondary amines.

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