The E isomer of (123)I-2beta-carbomethoxy-3beta-(4-fluorophenyl)-N-(1-iodoprop-1-en-3-yl)nortropane (Altropane(R)) shows high affinity (IC(50) = 6.62 +/- 0.78 nmol) and selectivity (DA/5-HT = 25) for DAT sites in the striatum. Recently, dynamic SPECT studies in healthy volunteers and patients with P
โฆ LIBER โฆ
A Highly Selective and Specific PET Tracer for Imaging of Tau Pathologies
โ Scribed by Zhang, Wei ;Arteaga, Janna ;Cashion, Daniel K. ;Chen, Gang ;Gangadharmath, Umesh ;Gomez, Luis F. ;Kasi, Dhanalakshmi ;Lam, Chung ;Liang, Qianwa ;Liu, Changhui ;Mocharla, Vani P. ;Mu, Fanrong ;Sinha, Anjana ;Szardenings, A. Katrin ;Wang, Eric ;Walsh, Joseph C. ;Xia, Chunfang ;Yu, Chul ;Zhao, Tieming ;Kolb, Hartmuth C.
- Book ID
- 118046443
- Publisher
- IOS Press
- Year
- 2012
- Tongue
- English
- Weight
- 998 KB
- Volume
- 31
- Category
- Article
- ISSN
- 1387-2877
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