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A convenient synthesis of tetrazole, precursors of α-dialkylated α-amino acids, by reaction of trimethylsilyl azide with α-dialkylated β-ketoesters

✍ Scribed by Henri-Jean Cristau; Xavier Marat; Jean-Pierre Vors; Jean-Luc Pirat

Book ID
104253308
Publisher
Elsevier Science
Year
2003
Tongue
French
Weight
132 KB
Volume
44
Category
Article
ISSN
0040-4039

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✦ Synopsis

The Schmidt rearrangement using trimethylsilyl azide with various a-dialkylated b-keto esters affords a convenient synthesis of tetrazole, precursors of a-dialkylated a-amino acids.

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