## Abstract A convenient synthesis of the antidepressant paroxetine starting from 1‐benzyl‐4‐piperidone (**2**) is reported. A stereoselective reduction resulted in __cis__‐piperidine‐3‐methanol [(**+**)‐**6**]. The reaction between __cis__‐piperidine‐3‐methanol mesylate (**7**) and sesamol led to
✦ LIBER ✦
A Convenient Synthesis of (-)-Paroxetine.
✍ Scribed by Laszlo Czibula; Andras Nemes; Ferenc Seboek; Csaba Jr. Szantay; Marianna Mak
- Publisher
- John Wiley and Sons
- Year
- 2004
- Weight
- 8 KB
- Volume
- 35
- Category
- Article
- ISSN
- 0931-7597
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