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A convenient preparation of 14C-labelled 5H-2,3-benzodiazepines

✍ Scribed by G. Zólyomi; T. Láng; J. Körösi; T. Hámori

Publisher
John Wiley and Sons
Year
1984
Tongue
French
Weight
331 KB
Volume
21
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

A convenient method for preparing 5__H__‐2,3‐benzodi‐azepines labelled with ^14^C was developed in which the corresponding phenylacetone derivatives were acylated by labelled aromatic carboxylic acid. In spite of the low yield, this method is advantageous in comparison the known ones because of the obtainable specific activity, which is a consequence of the few stages and simplicity of the synthesis.

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