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A concise route to tiazofurin

✍ Scribed by Richard S. Brown; James Dowden; Christelle Moreau; Barry V.L. Potter

Book ID
104251804
Publisher
Elsevier Science
Year
2002
Tongue
French
Weight
73 KB
Volume
43
Category
Article
ISSN
0040-4039

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✦ Synopsis

Successful oxidation of a key thiazoline intermediate allows an efficient synthesis of tiazofurin in four steps from commercially available 1%-acetoxy-2%,3%,5%-tri-O-benzoyl-b-D-ribofuranose.

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