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Tricyclic cephems as inhibitors of human leukocyte elastase. Furo[3,4-c]cepham sulfones

โœ Scribed by Marco Alpegiani; Pierluigi Bissolino; Riccardo Corigli; Vincenzo Rizzo; Ettore Perrone


Publisher
Elsevier Science
Year
1995
Tongue
English
Weight
182 KB
Volume
5
Category
Article
ISSN
0960-894X

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Design, synthesis and biological evaluat
โœ William C. Groutas; Michael J. Brubaker; Lee S. Chong; Radhika Venkataraman; He ๐Ÿ“‚ Article ๐Ÿ“… 1995 ๐Ÿ› Elsevier Science ๐ŸŒ English โš– 572 KB

Structure-activity relationship study and in vitro biochemical studies with human leukocyte elastase, cathepsin G and proteinase 3 were conducted using a series of succinimide derivatives.