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Traceless solid phase synthesis of 2,3-disubstituted indoles

✍ Scribed by Adrian L. Smith; Graeme I. Stevenson; Christopher J. Swain; JoséL. Castro

Publisher
Elsevier Science
Year
1998
Tongue
French
Weight
234 KB
Volume
39
Category
Article
ISSN
0040-4039

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✦ Synopsis

An efficient method for the traceless solid phase synthesis of 2,3-disubstituted indoles using a THP linker and a Pd(0)-mediated annulation of 2-iodoaniline and acetylenes is reported.

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