✦ LIBER ✦

The synthesis of novel GABA uptake inhibitors. Part 2. Synthesis of 5-hydroxytiagabine, a human metabolite of the GABA reuptake inhibitor tiagabine

✍ Scribed by Knud E. Andersen; Mikael Begtrup; Mukund S. Chorghade; Elaine C. Lee; Jesper Lau; Behrend F. Lundt; Hans Petersen; Per O. Sørensen; Henning Thøgersen

Publisher: Elsevier Science
Year: 1994
Tongue: French
Weight: 821 KB
Volume: 50
Category: Article
ISSN: 0040-4020
DOI: 10.1016/s0040-4020(01)85345-x

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

ChemInform Abstract: Synthesis of Novel

ChemInform Abstract: Synthesis of Novel γ-Aminobutyric Acid (GABA) Uptake Inhibitors. Part 5. Preparation and Structure—Activity Studies of Tricyclic Analogues of Known GABA Uptake Inhibitors.

✍ Knud Erik Andersen; Jan L. Soerensen; Jesper Lau; Behrend F. Lundt; Hans Peterse 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 34 KB 👁 1 views

Synthesis and Biochemical Studies of Spi

Synthesis and Biochemical Studies of Spirocyclic Amino Acid Esters, Part 3 Activity of 2-Azaspiro[4.5]decane-6-carboxylates as GABA-Uptake Inhibitors

✍ Wilhelm Fleischhacker; Silvia Lauritz; Ernst Urban; Peter Baumann; Helmut Bittig 📂 Article 📅 1996 🏛 John Wiley and Sons 🌐 English ⚖ 638 KB

ChemInform Abstract: A Novel Class of In

ChemInform Abstract: A Novel Class of Inhibitors for Human Steroid 5α-Reductase: Synthesis and Biological Evaluation of Indole Derivatives. Part 2.

✍ Susumu Igarashi; Hiroshi Inami; Hiromu Hara; Masahiro Fujii; Hiroshi Koutoku; Hi 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 32 KB 👁 1 views

ChemInform Abstract: Selective Inhibitor

ChemInform Abstract: Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues.

✍ Povl Krogsgaard-Larsen; et al. et al. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 36 KB 👁 2 views

ChemInform Abstract: Quaternary Substitu

ChemInform Abstract: Quaternary Substituted PDE IV Inhibitors. Part 2. The Synthesis and in vitro Evaluation of a Novel Series of γ-Lactams.

✍ C. HULME; K. MORIARTY; F.-C. HUANG; J. MASON; D. MCGARRY; R. LABAUDINIERE; J. SO 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 38 KB 👁 2 views

Synthesis of a novel α-glucoside of the

Synthesis of a novel α-glucoside of the powerful glucosidase inhibitor 2,5-dideoxy-2,5-imino-d-mannitol via enzymatic glucosylation of 5-azido-5-deoxy-d-fructopyranose

✍ Karl Dax; Michael Ebner; Roland Peinsipp; Arnold E. Stütz 📂 Article 📅 1997 🏛 Elsevier Science 🌐 French ⚖ 127 KB

Regio-and stereoselective enzymatic glucosylation of 5-azido-5-deoxy-D-fructopyranose with the aid of commerically available 0t-glucosidase from yeast allows easy access to the corresponding 4-O-~t-D-glucopyranosyl derivative of this non-natural ketose. This disaccharide gives, in one step, access t