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The first general synthesis of N-substituted 1,2-benzisoxazolin-3-ones

✍ Scribed by Guo-qiang Shi

Book ID: 104210050
Publisher: Elsevier Science
Year: 2000
Tongue: French
Weight: 163 KB
Volume: 41
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(00)00164-7

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✦ Synopsis

A convenient synthesis of the title compounds has been developed. Key synthetic steps include: (1) conversion of the readily available salicylic acid derivatives to the corresponding N-substituted salicylhydroxamic acids; (2) cyclization of the hydroxamic acids under Mitsunobu conditions to give the title compounds.

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