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The development of additional radioligands of varying pharmacokinetics for the 5-HT1A receptor

✍ Scribed by L. Lang; E. M. Jagoda; W. C. Eckelman

Book ID
112132538
Publisher
John Wiley and Sons
Year
2001
Tongue
French
Weight
148 KB
Volume
44
Category
Article
ISSN
0022-2135

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Synthesis of [3H]CP-93,129: A selective
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✍ John E Macor; Kevin Ryan; Phillip M. Chalabi; James C. Windels; Robert W. Roth 📂 Article 📅 1990 🏛 John Wiley and Sons 🌐 French ⚖ 413 KB

## Abstract The synthesis of [^3^H]‐CP‐93,129, a potent radioligand for the serotonin 5‐HT~1B~ receptor, is described. 5‐Butoxypyrrolo[3,2‐b]pyridine (2) is converted in 3 steps to 5‐butoxy‐1‐phenylsulfonyl‐2‐tritiopyrrolo[3,2‐b]pyridine (3c) via lithiation of C2, iodination of that anion, and trit