Aminoglycosides are among the most commonly used broadspectrum antibiotics. [1] The biological activity relies on their high affinity for the major groove of bacterial 16S rRNA, [2] thereby impeding protein synthesis. A number of aminoglycosides also display antiviral activity owing to specific inte
✦ LIBER ✦
Tethered Bisubstrate Derivatives as Probes for Mechanism and as Inhibitors of Aminoglycoside 3‘-Phosphotransferases
✍ Scribed by Liu, Meizheng; Haddad, Jalal; Azucena, Eduardo; Kotra, Lakshmi P.; Kirzhner, Maria; Mobashery, Shahriar
- Book ID
- 126770480
- Publisher
- American Chemical Society
- Year
- 2000
- Tongue
- English
- Weight
- 185 KB
- Volume
- 65
- Category
- Article
- ISSN
- 0022-3263
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