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Synthesis of the 6′-iso analogues of neplanocin A and 5′-homoneplanocin A

✍ Scribed by Wei Ye; Mingzhu He; Stewart W. Schneller

Publisher: Elsevier Science
Year: 2009
Tongue: French
Weight: 350 KB
Volume: 50
Category: Article
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2009.10.016

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✦ Synopsis

An efficient synthesis of 6'-isoneplanocin A and 6-isohomoneplanocin A is reported. The key steps in the synthesis include an enyne metathesis and a regioselective oxidation.

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