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Synthesis of radiolabelled photolabile fusidic acid analogues

✍ Scribed by Søren Christian Schou; Ditte Riber; Gunnar Grue-Sørensen

Publisher
John Wiley and Sons
Year
2007
Tongue
French
Weight
107 KB
Volume
50
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

Two analogues of the antibiotic fusidic acid with photolabile groups, 4‐azidophenyl and 4‐benzoylphenyl, were successfully labelled with tritium via Pd/C catalysed tritiation of unsaturated precursors. Specific activities of 36 and 44 Ci/mmol were obtained. Copyright © 2007 John Wiley & Sons, Ltd.

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