The t a r g e t compound, 1-([ Br1bromo)estradlol (la), was prepared i n t h r e e steps from 4-amlnoestradlol 3-methyl ether (2). E l e c t r o p h l l l c bromlnatlon o f 2 w l t h I n s l t u generated 7 7 B r C l f o l l o w e d by deamlnatlon I n t h e same r e a c t i o n m i x t u r e gave 1-
Synthesis of no-carrier-added radiobrominated N-alkylated analogues of spiperone
✍ Scribed by S. M. Moerlein; P. Laufer; G. Stöcklin
- Publisher
- John Wiley and Sons
- Year
- 1985
- Tongue
- French
- Weight
- 532 KB
- Volume
- 22
- Category
- Article
- ISSN
- 0022-2135
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