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Synthesis of five- and six-membered lactams via solvent-free microwave Ugi reaction

✍ Scribed by Mouhamad Jida; Sandra Malaquin; Rebecca Deprez-Poulain; Guillaume Laconde; Benoit Deprez

Book ID: 104098058
Publisher: Elsevier Science
Year: 2010
Tongue: French
Weight: 285 KB
Volume: 51
Category: Article
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2010.07.021

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✦ Synopsis

a b s t r a c t Five-and six-membered lactams were synthesized via a 4-center 3-component Ugi reaction by combining amines, isocyanides, and ketoacids under solvent-free microwave conditions. The reaction was carried out in much shorter times and the yields were improved in comparison to classical conditions.

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