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Synthesis of carbon-14 labeled clomiphene

✍ Scribed by P. Narasimha Rao; James W. Cessac

Publisher
John Wiley and Sons
Year
1985
Tongue
French
Weight
388 KB
Volume
22
Category
Article
ISSN
0022-2135

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✦ Synopsis

Clomiphene, 2-[4-(2-chloro-1,2-diphenylethenyl)phenoxy~-N.N- diethylethanamine, an antiestrogen, is a nonsteroidal triphenylethylene derivative. For the successful synthesis of carbon-14 labeled clomiphene it is essential to have a free radical inhibitor in the reaction medium.

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