Synthesis of 6(1-Methyl-4-nitro-5-|4,5-14 C| imidazolyl)thiopurinc (azathioprine)
β Scribed by Heather N. Yrowell; Gertrude B. Elion
- Book ID
- 112123079
- Publisher
- Journal of Heterocyclic Chemistry
- Year
- 1973
- Tongue
- English
- Weight
- 158 KB
- Volume
- 10
- Category
- Article
- ISSN
- 0022-152X
No coin nor oath required. For personal study only.
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## Abstract The increasing clinical importance of drugβresistant pathogens has lent additional urgency to antimicrobial research. Various 5β(1βmethylβ5βnitroβ2βimidazolyl)β4__H__β1, 2, 4βtriazoles (**4aβ6f**) were synthesized and tested __in vitro__ for their antibacterial and antifungal activities