✦ LIBER ✦

Synthesis of 3-(indol-2-yl)-propenoate derivatives of tryptamine, valuable intermediates for the preparation of indole alkaloids

✍ Scribed by Patrick D Bailey; Sean P Hollinshead

Book ID: 104227674
Publisher: Elsevier Science
Year: 1987
Tongue: French
Weight: 228 KB
Volume: 28
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(00)96233-6

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✦ Synopsis

~ A simple three step route to 3-(indol-2-yl)--propenoate derivatives of tryptamine has been developed, involving the base-induced ring-opening of protected tetrahydro-8-carbolines that result from a modified Pictet-Spengler reaction. Several recent syntheses of indole alkaloids have utilised Z-propenoate derivatives

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