✦ LIBER ✦

Synthesis of 2-[2-14C]-(2-aminoethyl)-thiazole dihydrochloride: Thiazolyl ethylamine dihydrochloride

✍ Scribed by M A Armitage; D Saunders

Publisher: John Wiley and Sons
Year: 1985
Tongue: French
Weight: 182 KB
Volume: 22
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580221010

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✦ Synopsis

The hlstamlne H1 agonlst, 2-[2-14C]-(2-amlnoethyl)-thlazole dlhydrochlorlde has been l a b e l l e d w t t h carbon-14 I n the 2 p o s l t l o n of the t h l a z o l e s t a r t l n g from potasslum [14C] cyanlde. The o v e r a l l radlochemlcal y i e l d f o r the synthesls was 17% a t a s p e c i f i c a c t i v i t y o f 36mCl/m01.

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