✦ LIBER ✦

Synthesis and Structure−Activity Relationships of Truncated Bisubstrate Inhibitors of Aminoglycoside 6‘- N -Acetyltransferases

✍ Scribed by Gao, Feng; Yan, Xuxu; Shakya, Tushar; Baettig, Oliver M.; Ait-Mohand-Brunet, Samia; Berghuis, Albert M.; Wright, Gerard D.; Auclair, Karine

Book ID: 121464353
Publisher: American Chemical Society
Year: 2006
Tongue: English
Weight: 145 KB
Volume: 49
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm060732n

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Regio- and Chemoselective 6′-N-Derivatiz

Regio- and Chemoselective 6′-N-Derivatization of Aminoglycosides: Bisubstrate Inhibitors as Probes To Study Aminoglycoside 6′-N-Acetyltransferases

✍ Feng Gao; Xuxu Yan; Oliver M. Baettig; Albert M. Berghuis; Karine Auclair 📂 Article 📅 2005 🏛 John Wiley and Sons 🌐 English ⚖ 141 KB

Aminoglycosides are among the most commonly used broadspectrum antibiotics. [1] The biological activity relies on their high affinity for the major groove of bacterial 16S rRNA, [2] thereby impeding protein synthesis. A number of aminoglycosides also display antiviral activity owing to specific inte

Regio- and Chemoselective 6′-N-Derivatiz

Regio- and Chemoselective 6′-N-Derivatization of Aminoglycosides: Bisubstrate Inhibitors as Probes To Study Aminoglycoside 6′-N-Acetyltransferases

✍ Feng Gao; Xuxu Yan; Oliver M. Baettig; Albert M. Berghuis; Karine Auclair 📂 Article 📅 2005 🏛 John Wiley and Sons 🌐 English ⚖ 142 KB

Synthesis of 4′-aminopantetheine and der

Synthesis of 4′-aminopantetheine and derivatives to probe aminoglycoside N-6′-acetyltransferase

✍ Yan, Xuxu; Akinnusi, T. Olukayode; Larsen, Aaron T.; Auclair, Karine 📂 Article 📅 2011 🏛 Royal Society of Chemistry 🌐 English ⚖ 398 KB

Synthesis and structure-activity relatio

Synthesis and structure-activity relationships of new ACAT inhibitors

✍ JY Nioche; J Decerprit; D Festal 📂 Article 📅 1995 🏛 Elsevier Science 🌐 French ⚖ 732 KB

Structure-activity relationships for sub

Structure-activity relationships for substrates and inhibitors of pineal 5-hydroxytryptamine-N-acetyltransferase: preliminary studies

✍ Shuren Shen; Béatrice Brémont; Isabelle Serraz; Jean Andrieux; Annie Poncet; Mon 📂 Article 📅 1996 🏛 Elsevier Science 🌐 English ⚖ 988 KB

Novel acetylcholinesterase inhibitors: S

Novel acetylcholinesterase inhibitors: Synthesis and structure–activity relationships of phthalimide alkyloxyphenyl N,N-dimethylcarbamate derivatives

✍ Qianfei Zhao; Guoquan Yang; Xiangdong Mei; Huizhu Yuan; Jun Ning 📂 Article 📅 2009 🏛 Elsevier Science 🌐 English ⚖ 225 KB