The syntheses of the thiophenic analogue of Moprolol (Id) and of its related compound l a are described. From a preliminary pharmacological evaluation compound Id seems worthy of further studies due to its notable P-blocking activity and its remarkable anti-platelet aggregation action. ## Synthese
✦ LIBER ✦
Synthesis and Preliminary Pharmacological Study of Thiophene Analogues of the Antipyretic and Analgesic Agent Ethenzamide
✍ Scribed by V. Darias; L. Bravo; S. S. Abdallah; C. C. Sánchez Mateo; M. A. Expósito-orta; J. Lissavetsky; J. Manzanares
- Publisher
- John Wiley and Sons
- Year
- 1992
- Tongue
- English
- Weight
- 381 KB
- Volume
- 325
- Category
- Article
- ISSN
- 0365-6233
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