5'-Ester derivatives of the potent adenosine agonists N6-[4-[[[[4-[[[(2-acetylaminoethyl)amino]carbonyl]methyl] anilino]carbonyl]methyl]phenyl]adenosine (N-AcADAC; 1) and N6-cyclopentyladenosine (CPA; 2) were prepared as prodrugs. Both alkyl esters or carbonates (designed to enter the brain by virtu
✦ LIBER ✦
Synthesis and biological activities of peptidomimetic analogues of compound A71623, a potent and selective CCK-A receptor agonist
✍ Scribed by Jean-Christophe Califano; Laurent Goullieux; Muriel Amblard; Jean-Alain Fehrentz; Nicole Bernad; Gilbert Bergé; Jean Castel; Jean Martinez
- Publisher
- Springer Netherlands
- Year
- 1997
- Tongue
- English
- Weight
- 274 KB
- Volume
- 4
- Category
- Article
- ISSN
- 1573-3149
No coin nor oath required. For personal study only.
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