Bioisosteric Modification of Salvinorin A, a Potent and Selective ϰ-Opioid Receptor Agonist.

Asymmetric Synthesis of Salvinorin A (I)

Asymmetric Synthesis of Salvinorin A (I), a Potent ϰ Opioid Receptor Agonist.

✍ Jonathan R. Scheerer; Jonathan F. Lawrence; Grace C. Wang; David A. Evans 📂 Article 📅 2007 🏛 John Wiley and Sons ⚖ 14 KB

A Highly Selective ϰ-Opioid Receptor Ago

A Highly Selective ϰ-Opioid Receptor Agonist with Low Addictive Potential and Dependence Liability.

✍ Hee Sock Park; Hee Yoon Lee; Yong Hae Kim; Jin Kyu Park; Edwin E. Zvartau; Heese 📂 Article 📅 2006 🏛 John Wiley and Sons ⚖ 12 KB

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.

Synthesis of [3H]DIPPA: A potent irrever

Synthesis of [3H]DIPPA: A potent irreversible antagonist selective for the κ opioid receptor

✍ An-Chih Chang; Joseph D. Trometer; Philip S. Portoghese 📂 Article 📅 1995 🏛 John Wiley and Sons 🌐 French ⚖ 222 KB

## Abstract 2‐(3,4‐Dichlorophenyl)‐N‐methyl‐N‐[(1S)‐1‐(3‐isothiocyanatophenyl)‐2‐(1‐pyrrolidinyl)ethyl]acetamide (1, DIPPA) has been previously reported to be an opioid receptor affinity label that produces selective and long‐lasting κ opioid receptor antagonism in mice, High specific activity [^3^

Azepinone as a Conformational Constraint

Azepinone as a Conformational Constraint in the Design of ϰ-Opioid Receptor Agonists.

✍ Roland E. Dolle; et al. et al. 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 23 KB

## Abstract For Abstract see ChemInform Abstract in Full Text.

Highly Potent and Selective Zwitterionic

Highly Potent and Selective Zwitterionic Agonists of the δ-Opioid Receptor. Part 1.

✍ Donald S. Middleton; Graham N. Maw; Clare Challenger; Alan Jessiman; Patrick S. 📂 Article 📅 2006 🏛 John Wiley and Sons ⚖ 20 KB

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.

Syntheses of 10-Oxo, 10α-Hydroxy, and 10

Syntheses of 10-Oxo, 10α-Hydroxy, and 10β-Hydroxy Derivatives of a Potent ϰ-Opioid Receptor Agonist, TRK-820.

✍ Hiromasa Horikiri; Noriyuki Hirano; Yoichiro Tanaka; Junji Oishi; Hitoshi Hatake 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 28 KB

## Abstract For Abstract see ChemInform Abstract in Full Text.