✦ LIBER ✦

Synthesis and analgesic properties of some conformationally restricted analogs of profadol

✍ Scribed by Crooks, Peter A.; Szyndler, Richard

Book ID: 126188687
Publisher: American Chemical Society
Year: 1980
Tongue: English
Weight: 484 KB
Volume: 23
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm00180a021

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis of some conformationally restr

Synthesis of some conformationally restricted analogs of fentanyl

✍ Berger, Joel G.; Davidson, Fredric; Langford, Gordon E. 📂 Article 📅 1977 🏛 American Chemical Society 🌐 English ⚖ 397 KB

Conformationally restricted leukotriene

Conformationally restricted leukotriene antagonists. Stereoselective synthesis of some leukotriene D4 analogs

✍ Jeffrey S. Sabol; Philip M. Weintraub; Thomas H. Gieske; Robert J. Cregge 📂 Article 📅 1990 🏛 Elsevier Science 🌐 French ⚖ 385 KB

The stereocontrolled synthesis of conformationally restricted LTD4 analogs 2a. b is described. Epoxidation of enone 4 affords a 2.4:1 mixture of trans-epoxide 5 and cis-epoxide 9. Stereocontrolled elaboration of each epoxide to final product involves stereoselective Wittig olefination to Z-olefins 6

Synthesis of (+)- and (−)-milnaciprans a

Synthesis of (+)- and (−)-milnaciprans and their conformationally restricted analogs

✍ Satoshi Shuto; Shizuka Ono; Yukako Hase; Noriko Kamiyama; Akira Matsuda 📂 Article 📅 1996 🏛 Elsevier Science 🌐 French ⚖ 236 KB

Stereocontrolled syntheses of some confo

Stereocontrolled syntheses of some conformationally restricted analogs of serotonin

✍ Arun Ghosh; Wuyi Wang; Jeremiah P. Freeman; John S. Althaust; Philip F. VonVoigt 📂 Article 📅 1991 🏛 Elsevier Science 🌐 French ⚖ 659 KB

The synthesis and analgesic activities o

The synthesis and analgesic activities of some spiro[indan-1,3′-pyrrolidine] derivatives designed as rigid analogs of profadol

✍ P. A. Crooks; R. Sommerville 📂 Article 📅 1982 🏛 John Wiley and Sons 🌐 English ⚖ 453 KB

Conformationally restricted leukotriene

Conformationally restricted leukotriene antagonists. Asymmetric synthesis of some nor-leukotriene D4 analogs

✍ Jeffrey S Sabol; Robert J Cregge 📂 Article 📅 1989 🏛 Elsevier Science 🌐 French ⚖ 167 KB

The enantiomeric pair of conformationally-restricted nor-LTD4 analogs s and 11 have been synthesized stereoselectively from (g)-2-cyclohexen-l-01. Due to our continuing interest in the stereoselective syntheses of conformationallyrestricted LTDl analogsr, we were attracted by recent reports' that 2-