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Structural and ionic determinants of 5-nitro-2-(3-phenylpropylamino)-benzoic acid block of the CFTR chloride channel

โœ Scribed by Kenneth B Walsh; Kathryn J Long; Xufeng Shen


Book ID
110004310
Publisher
Nature Publishing Group
Year
1999
Tongue
English
Weight
188 KB
Volume
127
Category
Article
ISSN
0007-1188

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5-Nitro-2-(3-phenylpropylamino)benzoic acid (NPPB) has been shown to produce a reduction in channel open probability in a number of epithelial chloride channels. We have investigated its action on a calcium-dependent airway epithelial chloride channel, which shows voltage-dependent gating following