๐”– Bobbio Scriptorium
โœฆ   LIBER   โœฆ

Solid Support Synthesis of Tetrahydroquinolines via the Grieco Three Component Condensation

โœ Scribed by Alexander S. Kiselyov; Robert W. Armstrong

Book ID
104257772
Publisher
Elsevier Science
Year
1997
Tongue
French
Weight
493 KB
Volume
38
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.

๐Ÿ“œ SIMILAR VOLUMES

Solid support synthesis of polysubstitut
Solid support synthesis of polysubstituted tetrahydroquinolines via three-component condensation catalyzed by Yb(OTf)3
โœ Alexander S. Kiselyov; Leon Smith II; Robert W. Armstrong ๐Ÿ“‚ Article ๐Ÿ“… 1998 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 469 KB

Solid support synthesis of polysubstituted tetrahydroquinolines is described. The procedure is based on a three-component condensation involving immobilized derivatives of 4-aminophenylalanine, aldehydes, alkenes and Yb(OTf) 3 as a catalyst. The methodology is further expanded to the solid support s

Solid-phase synthesis of 4-aryl-1,4-dihy
Solid-phase synthesis of 4-aryl-1,4-dihydropyridines via the Hantzsch three component condensation
โœ J.Guy Breitenbucher; Gina Figliozzi ๐Ÿ“‚ Article ๐Ÿ“… 2000 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 159 KB

We report the synthesis of 1,4-dihydropyridines on solid support utilizing the Hantzsch condensation. Unwanted reactive impurities were removed from the desired products, by selective cleavage from solid support. The synthesis of a 272 compound library is reported using the methods described.