✦ LIBER ✦

Solid-phase synthesis of N-substituted 3,4-dihydroquinazolinone derivatives

✍ Scribed by Zhang Liu; Lili Ou; Marc A. Giulianotti; Richard A. Houghten

Publisher: Elsevier Science
Year: 2011
Tongue: French
Weight: 198 KB
Volume: 52
Category: Article
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2011.03.034

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✦ Synopsis

An efficient solid-phase synthetic approach for the synthesis of N-substituted 3, 4-dihydroquinazolinone derivatives has been developed. Four different 2-nitrobenzoic acids and three different 2-phenylacetyl chlorides were employed in the synthesis of this library. After purification, all products were obtained in good yields.

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