𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Solid-Phase Synthesis of a 4-Substituted γ-Lactam Library

✍ Scribed by Vergnon, Anne L.; Pottorf, Richard S.; Winters, Michael P.; Player, Mark R.


Book ID
126051487
Publisher
American Chemical Society
Year
2004
Tongue
English
Weight
229 KB
Volume
6
Category
Article
ISSN
1520-4766

No coin nor oath required. For personal study only.


📜 SIMILAR VOLUMES


γ-Methyl-substituted-γ-butyrolactones: s
✍ Nicolas Gouault; Jean-François Cupif; Armelle Sauleau; Michèle David 📂 Article 📅 2000 🏛 Elsevier Science 🌐 French ⚖ 163 KB

The solid-phase synthesis of several g-methyl-substituted-g-butyrolactones using a cyclisation±cleavage reaction is reported. Chemical modi®cations of polymer-bound azido (2a) and iodo alcohols (2b) were realised in order to introduce additional diversity onto the lactone structure.

Solid-phase synthesis of 2-substituted-3
✍ Shingo Makino; Tatsuya Okuzumi; Eiji Nakanishi; Takashi Tsuji 📂 Article 📅 2002 🏛 Elsevier Science 🌐 French ⚖ 91 KB

The first solid-phase synthesis of 2-substituted-3-(substituted sulfanyl)-1,2,4-benzothiadiazine 1,1-dioxides has been developed. Synthesis of the title compounds was achieved as follows: (1) sulfonylation of solid-supported primary amines with 2-nitrobenzenesulfonylchlorides, (2) reduction of the n

Solid-phase synthesis of γ-lactams, γ-la
✍ Richard C.D Brown; John Keily; Rehana Karim 📂 Article 📅 2000 🏛 Elsevier Science 🌐 French ⚖ 171 KB

Resin-bound cyclobutanone iminium salts, prepared on the solid-phase using the [2+2]-keteneiminium olefin cycloaddition reaction, have been transformed into a number of distinct structural classes including γ-lactams, γ-lactones, cyclobutylamines and cyclobutanols.