Following up on the observation that the dynorphin analog [Pro(3)]Dyn A(1-11)-NH(2) 2 possesses high affinity and selectivity for the kappa opioid receptor, a number of related peptides were prepared and characterized by radioligand binding and [(35)S]GTPgammaS assays. While incorporation of 2-azeti
Relationship between the Structure and Antimycobacterial Activity of Substituted Salicylanilides
✍ Scribed by Karel Waisser; Otakar Bureš; Pavel Holý; Jiří Kuneš; Radek Oswald; Lucie Jirásková; Milan Pour; Věra Klimešová; Lenka Kubicová; Jarmila Kaustová
- Publisher
- John Wiley and Sons
- Year
- 2003
- Tongue
- English
- Weight
- 152 KB
- Volume
- 336
- Category
- Article
- ISSN
- 0365-6233
No coin nor oath required. For personal study only.
📜 SIMILAR VOLUMES
## Abstract Enzymes are attractive catalysts for the production of optically active compounds in organic solvents. However, their often low catalytic activity in such applications hampers their practical use. To overcome this, we investigated the effectiveness of the covalent modification of α‐chym
A series of 2-amino-5-substituted pyridine derivatives was synthesized and their molluscicidal activity against white garden, Theba pisana (Mu È ller), and brown garden, Helix aspersa (Mu È ller), snails was investigated by two methods of application. Some of these compounds showed strong activity u