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Radioimmunoassay for imidapril, a new angiotensin-converting enzyme inhibitor, and imidaprilat, its active metabolite, in human plasma and urine

✍ Scribed by Kenta Yamanaka; Shigeki Morikawa; Kazuo Murata; Kiyoshi Banno; Tadashi Sato; Tsutomu Takai; Takchiko Suzuki; Masakazu Mizobe; Masao Ito; Kaichiro Ishibashi


Publisher
Elsevier Science
Year
1996
Tongue
English
Weight
447 KB
Volume
14
Category
Article
ISSN
0731-7085

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The disposition characteristics of pentopril (the ethyl ester) and its active carboxylic acid metabolite (CGS 13934) were determined in conscious rats after separate intravenous administrations of both compounds. The relationship between plasma concentration and pharmacological effect was also evalu