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Preparation of pyridyl grignard reagents and cross coupling reactions with sulfoxides bearing azaheterocycles

โœ Scribed by Naomichi Furukawa; Tadao Shibutani; Hisashi Fujihara

Publisher
Elsevier Science
Year
1987
Tongue
French
Weight
240 KB
Volume
28
Category
Article
ISSN
0040-4039

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โœฆ Synopsis

Pyridyl Grignard reagents were prepared from the corresponding iodopyridine and EtMgBr. New cross coupling reactions of the Grignard reagents with azaheterocycles took place on the sulfinyl sulfur atom to afford biazaheteroaryls.

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