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Preparation of 6-azaoxindole (6-azaindol-2(3H)-one) and substituted derivatives

✍ Scribed by Einar J. Andreassen; Jan M. Bakke

Publisher
Journal of Heterocyclic Chemistry
Year
2006
Tongue
English
Weight
105 KB
Volume
43
Category
Article
ISSN
0022-152X

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✦ Synopsis

Abstract

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A general synthesis of 6‐azaoxindoles, substituted in the 3‐ and 5‐position, has been developed starting from 4‐methoxycarbomethyl‐3‐nitropyridine, via hydrogenation of the nitro group and cyclisation of the resulting 3‐amino‐4‐methoxycarbomethyl‐pyridine.

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