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Potential drugs labelled with 14C. II. Synthesis of 1-cyano-3-imino-8, 9-dimethoxy-3, 4,5,6- -tetrahydro-thiazolo[4, 3-a]isoquinoline hydrochloride

✍ Scribed by E. Koltai; G. Zólyomi; P. Komáromy; D. Bánfi; T. Szüts; K. Takács

Publisher
John Wiley and Sons
Year
1981
Tongue
French
Weight
295 KB
Volume
18
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

The synthesis of 1‐cyano‐3‐imino‐8,9‐dimethoxy‐ ‐3,4, 5,6‐tetrahydro‐thiazolo [4,3‐a]isoquinoline hydrochloride labelled with ^14^C in five different positions: in position 3 (1a), in the cyano group at position 1 (1b), in position 5 (1c), in position 10b (1d) and in the methoxy groups at position 8 and 9 (1e) was carried out.

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