Synthesis of A-79175: a second generatio
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Daniel A. Dickman; Yi-Yin Ku; Howard E. Morton; Sanjay R. Chemburkar; Hemantkuma
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Article
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1997
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Elsevier Science
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English
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A convergent, high yielding, and scalable synthesis of A-79175, with a key step involving a mild and efficient Cu-Pd catalyzed coupling reaction of a terminal acetylene with a substituted 2-iodofuran is discussed.