𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Opioid peptides. Synthesis and biological properties of dermorphin related hexapeptides

✍ Scribed by Severo Salvadori; Mauro Marastoni; Gianfranco Balboni; Pierandrea Borea; Roberto Tomatis

Publisher
Elsevier Science
Year
1990
Tongue
French
Weight
775 KB
Volume
25
Category
Article
ISSN
0223-5234

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis and biological activity of hom
Synthesis and biological activity of homoarginine-containing opioid peptides
✍ Jan Izdebski; Danuta Kunce; Peter W. Schiller; Nga N. Chung; Tomasz Gers; Monika 📂 Article 📅 2006 🏛 John Wiley and Sons 🌐 English ⚖ 93 KB

## Abstract Two tris‐alkoxycarbonyl homoarginine derivatives, Boc‐Har{ω,ω′‐[Z(2Br)]~2~}‐OH and Boc‐Har{ω,ω′‐[Z(2Cl)]~2~}‐OH, were prepared by guanidinylation of Boc‐Lys‐OH, and used for the synthesis of neo‐endorphins and dynorphins. The results were compared with that obtained in the synthesis in

Synthesis and Biological Properties of E
Synthesis and Biological Properties of Enkephalin-like Peptides Containing Carboranylalanine in Place of Phenylalanine
✍ Robert Schwyzer; Kim Quang Do; Alex N. Eberle; Jean-Luc Fauchére 📂 Article 📅 1981 🏛 John Wiley and Sons 🌐 German ⚖ 421 KB

## Abstract The syntheses of [D‐Ala^2^, Car^4^, Leu^5^]‐enkephalin, its amide, and of [D‐Ala^2^, Car^4^, Met^5^]‐enkephalin amide are described in detail. The three compounds show pronounced morphine‐like potencies in certain bio‐assays, and were used to investigate the influence of electronic, ste

Synthesis and Biological Properties of E
Synthesis and Biological Properties of Enkephalin-like Peptides Containing Adamantylalanine in Position 4 and 5
✍ Kim Quang Do; Robert Schwyzer 📂 Article 📅 1981 🏛 John Wiley and Sons 🌐 German ⚖ 356 KB

## Abstract The syntheses of seven [D‐ala‐^2^]‐enkephalin analogues, H‐Tyr‐ala‐Gly‐X‐Y, with X‐Y = Phe‐Ada‐OH, Phe‐ada‐OH, Phe‐Ada‐NH~2~, Phe‐ada‐NH~2~, Ada‐Leu‐OH, Ada‐Leu‐NH~2~, and Ada‐Ada‐NH~2~ are described. The compounds with Y = Ada (= L‐Ada) or ada (= D‐Ada) show pronounced morphine‐like ac

Synthesis and properties of the first al
Synthesis and properties of the first all-aza analogue of a biologically active peptide
✍ Prof. Dr. Joachim Gante; Michael Krug; Günter Lauterbach; Reinhard Weitzel; W. H 📂 Article 📅 1995 🏛 John Wiley and Sons 🌐 English ⚖ 370 KB

The synthesis of the first all-aza-amino acid analogue (2) of a peptidic renin inhibitor is described. The X-ray structural analysis and molecular modelling investigations of this novel compound reveal interesting conformational features which have a significant impact on its biological activity. In