New antitumour cyclic astin analogues: synthesis, conformation and bioactivity
✍ Scribed by Dr Filomena Rossi; Giancarlo Zanotti; Michele Saviano; Rosa Iacovino; Pasquale Palladino; Gabriella Saviano; Pietro Amodeo; Teodorico Tancredi; Paolo Laccetti; Catherine Corbier; Ettore Benedetti
- Book ID
- 105360320
- Publisher
- John Wiley and Sons
- Year
- 2004
- Tongue
- English
- Weight
- 170 KB
- Volume
- 10
- Category
- Article
- ISSN
- 1075-2617
- DOI
- 10.1002/psc.506
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📜 SIMILAR VOLUMES
## Abstract We synthesized by solution‐phase methods three analogues, [L‐Leu^6^‐OMe], [L‐(αMe)Leu^3^, L‐Leu^6^‐OMe], and [L‐(αMe)Val^4^, L‐Leu^6^‐OMe] of halovir A. The [L‐Leu^6^‐OMe] analogue is known to be biologically equipotent to its naturally occurring, antiviral, lipopentapeptide amide paren
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