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N -Hydroxy-3-phenyl-2-propenamides as Novel Inhibitors of Human Histone Deacetylase with in Vivo Antitumor Activity: Discovery of (2 E )- N -Hydroxy-3-[4-[[(2-hydroxyethyl)[2-(1 H -indol-3-yl)ethyl]amino]methyl]phenyl]-2-propenamide (NVP-LAQ824)

✍ Scribed by Remiszewski, Stacy W.; Sambucetti, Lidia C.; Bair, Kenneth W.; Bontempo, John; Cesarz, David; Chandramouli, Nagarajan; Chen, Ru; Cheung, Min; Cornell-Kennon, Susan; Dean, Karl; Diamantidis, George; France, Dennis; Green, Michael A.; Howell, Kobporn Lulu; Kashi, Rina; Kwon, Paul; Lassota, Peter; Martin, Mary S.; Mou, Yin; Perez, Lawrence B.; Sharma, Sushil; Smith, Troy; Sorensen, Eric; Taplin, Francis; Trogani, Nancy; Versace, Richard; Walker, Heather; Weltchek-Engler, Susan; Wood, Alexander; Wu, Arthur; Atadja, Peter

Book ID: 121012479
Publisher: American Chemical Society
Year: 2003
Tongue: English
Weight: 284 KB
Volume: 46
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm030235w

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