Interaction of 3,8-diazabicyclo (3.2.1) octanes with mu and delta opioid receptors
โ Scribed by G. Cignarella; D. Barlocco; M.E. Tranquillini; A. Volterra; N. Brunello; G. Racagni
- Book ID
- 114075309
- Publisher
- Elsevier Science
- Year
- 1988
- Weight
- 460 KB
- Volume
- 20
- Category
- Article
- ISSN
- 0031-6989
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A series of trimethyipiperazine derivatives, structurally related to the Ix-agonist 3-cinnamyl-8-propionyl-3,8-diazabicyclo[3.2.1]octane, have been synthesized and teswxl in binding studies, using 3H-DAMGO as Ix-selective ligand. Their different affinity towards Ix-opioid receptors has been interpre