Ketanserin. 3-~2-~4-~4-fluorobenzoyl~-l-piperidinyllethyll-2,4(1H,3H)-quinazol- inedione is a new serotonin S2-receptor blocking agent used in hypertension and related diseases. Pharmacokinetic studies required the synthesis of monolabelled 3H-and 14C-ketanserin tartrate. The tritium compound had th
Enzymic synthesis of lactose-14C (galactosyl-14C) and lactose-3H (glucosyl-3H)
β Scribed by B.G. Hudson; L. McKenzie; K.E. Ebner
- Publisher
- Elsevier Science
- Year
- 1972
- Tongue
- English
- Weight
- 292 KB
- Volume
- 48
- Category
- Article
- ISSN
- 0003-2697
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β¦ Synopsis
Recent enzymic studies Cl-3j have shown that, lactose is synthesized in the presence of substrates, a galactosyltjransferasc and a-lactalbumin. The reaction (equat'ion 1) is essentially irreversible and conditions may Rills+ 'Journal Article 2461 of the Agricultural Experiment Station,
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