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Efficient Synthesis of 1,4-Thiazepin-3-one Derivatives and Their Ring Transformations

✍ Scribed by Zaleska, Barbara ;Cież, Dariusz ;Grochowski, Jacek ;Serda, Pawel ;Winnik, Witold

Publisher
John Wiley and Sons
Year
2006
Tongue
English
Weight
535 KB
Volume
1996
Category
Article
ISSN
0947-3440

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✦ Synopsis

Abstract

A new one‐pot synthesis of title compounds 2 by reaction of β‐aminothiocinnamic acid anilides 1 with α‐haloacid halides is described. The ring of 1,4‐thiazepine 2 in basic medium undergoes transformation to thiazolidin‐4‐ones 5.

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