✦ LIBER ✦

Efficient and tunable synthesis of new polydentate bifunctional chelating agents using click chemistry

✍ Scribed by Clément Camp; Sandra Dorbes; Claude Picard; Eric Benoist

Book ID: 108284837
Publisher: Elsevier Science
Year: 2008
Tongue: French
Weight: 128 KB
Volume: 49
Category: Article
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2008.01.086

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis of Small Peptides and Their Us

Synthesis of Small Peptides and Their Use as Bifunctional Chelating Agents in Diagnostic Radiopharmaceuticals

✍ Chongzhi TANG; Longjin LI; Zhen PANG; Zhibin YUAN 📂 Article 📅 2009 🏛 John Wiley and Sons 🌐 English ⚖ 295 KB 👁 1 views

## Abstract Three linear mercaptoacetyl tetrapeptides, MAG3‐Leu‐OH, MAG3‐Phe‐OH and MAG3‐Tyr‐OH, were synthesized via a liquid phase synthetic approach with high yields and high purities without using preparative HPLC technique. The obtained products could be radiolabeled easily with ^99m^Tc under

Synthesis and evaluation of a macrocycli

Synthesis and evaluation of a macrocyclic bifunctional chelating agent for use with bismuth radionuclides

✍ K Garmestani; Z Yao; M Zhang; K Wong; C.W Park; I Pastan; J.A Carrasquillo; M.W 📂 Article 📅 2001 🏛 Elsevier Science 🌐 English ⚖ 205 KB

ChemInform Abstract: Synthesis of a New

ChemInform Abstract: Synthesis of a New Class of Isothiocyanatopeptide Bifunctional Chelating Agents for Coupling to Monoclonal Antibodies.

✍ S. RAM; D. J. BUCHSBAUM 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 31 KB

Synthesis, docking and in vitro antimala

Synthesis, docking and in vitro antimalarial evaluation of bifunctional hybrids derived from β-lactams and 7-chloroquinoline using click chemistry

✍ Pardeep Singh; Parvesh Singh; Malkeet Kumar; Jiri Gut; Philip J. Rosenthal; Kewa 📂 Article 📅 2012 🏛 Elsevier Science 🌐 English ⚖ 742 KB

Synthesis and evaluation of a new bifunc

Synthesis and evaluation of a new bifunctional chelating agent for 99mTc labeling proteins: p-carboxyethylphenylglyoxal-di(N-methylthiosemicarbazone)

✍ Arano, Yasushi; Yokoyama, Akira; Magata, Yasuhiro; Saji, Hideo; Horiuchi, Kazuko 📂 Article 📅 1986 🏛 Elsevier Science ⚖ 482 KB

A simple and efficient synthesis of a de

A simple and efficient synthesis of a derivatized pseudotripeptide containing a methylene thioether isostere and its use for the design of bifunctional rhenium and technetium chelating agents

✍ Matthias Scheunemann; Bernd Johannsen 📂 Article 📅 1997 🏛 Elsevier Science 🌐 French ⚖ 129 KB

A new approach to a pseudotripeptide based tetradentate chelating unit functionalizable with various bioactive groups has been developed. Using a one-pot reaction, a given 0)-aminoalkyl compound has been converted to a methylene thioether peptide isostere by two consecutive ring opening reactions.