The synthesis of a library of homoallylic amines is reported. The key step in the synthesis is a one-pot Nacyliminium ion coupling involving a solid phase-bound carbamate, an aldehyde and an allylsilane under Lewis acid conditions.
β¦ LIBER β¦
Efficiencies of reductive amination reactions on different solid supports
β Scribed by Chinh T. Bui; Firas A. Rasoul; Francesca Ercole; Yen Pham; N.Joe Maeji
- Book ID
- 108387183
- Publisher
- Elsevier Science
- Year
- 1998
- Tongue
- French
- Weight
- 238 KB
- Volume
- 39
- Category
- Article
- ISSN
- 0040-4039
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