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Discovery, Optimization, and Biological Evaluation of 5-(2-(Trifluoromethyl)phenyl)indazoles as a Novel Class of Transient Receptor Potential A1 (TRPA1) Antagonists

✍ Scribed by Rooney, Lisa; Vidal, Agnès; D’Souza, Anne-Marie; Devereux, Nick; Masick, Brian; Boissel, Valerie; West, Ryan; Head, Victoria; Stringer, Rowan; Lao, Jianmin; Petrus, Matt J.; Patapoutian, Ardem; Nash, Mark; Stoakley, Natalie; Panesar, Moh; Verkuyl, J. Martin; Schumacher, Andrew M.; Petrassi, H. Michael; Tully, David C.

Book ID: 124065094
Publisher: American Chemical Society
Year: 2014
Tongue: English
Weight: 807 KB
Volume: 57
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm401986p

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