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Discovery of an Orally Bioavailable NK1 Receptor Antagonist, (2S,3S)-(2-Methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with Potent Antiemetic Activity

✍ Scribed by Ward, Peter; Armour, Duncan R.; Bays, David E.; Evans, Brian; Giblin, Gerard M. P.; Heron, Nicola; Hubbard, Tania; Liang, Kai; Middlemiss, David

Book ID: 121231165
Publisher: American Chemical Society
Year: 1995
Tongue: English
Weight: 964 KB
Volume: 38
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm00026a005

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