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Discovery of 1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-2-imidazolidinone (GSK163090), a Potent, Selective, and Orally Active 5-HT 1A/B/D Receptor Antagonist

✍ Scribed by Leslie, Colin P.; Biagetti, Matteo; Bison, Silvia; Bromidge, Steven M.; Di Fabio, Romano; Donati, Daniele; Falchi, Alessandro; Garnier, Martine J.; Jaxa-Chamiec, Albert; Manchee, Gary; Merlo, Giancarlo; Pizzi, Domenica A.; Stasi, Luigi P.; Tibasco, Jessica; Vong, Antonio; Ward, Simon E.; Zonzini, Laura

Book ID: 118143907
Publisher: American Chemical Society
Year: 2010
Tongue: English
Weight: 896 KB
Volume: 53
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm100714c

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